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ScreeNingBio's GPCR Solution:
Assay Designed to Reach Your Goal Faster

​​Comprehensive GPCR Coverage

  • Ready-to use stable cell lines covering 80% GPCR drug targets

Native Expression Advantage

  • Full-length GPCRs stably expressed without artificial tags to preserve native receptor pharmacology

Flexible Assay Readouts

  • Multiple assay formats available, including cAMP, calcium flux, β-arrestin recruitment, IP-One, and reporter gene readouts, to meet diverse discovery needs

Cross-Species Capabilities

  • Broad panel of human, mouse, rat, dog, and cynomolgus monkey targets available for translational research

GPCR Family Tree.jpg
Target Receptors
按 类别-Target Receptors 篩選
Species
按 类别-Species 篩選
Assay Mode
按 类别-Assay Mode 篩選
Parental Line
按 类别-Receptor Form 篩選
CHO-K1/Mouse MT2 Stable Cell

SPECIES: Mouse

TARGET FAMILY: MT2 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0148B


CHO-K1/Rat MT2 Stable Cell

SPECIES: Rat

TARGET FAMILY: MT2 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0148C


CHO-K1/Human mGlu2 Stable Cell

SPECIES: Human

TARGET FAMILY: mGlu2 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0150A


CHO-K1/Human mGlu6 Stable Cell

SPECIES: Human

TARGET FAMILY: mGlu6 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0154A


CHO-K1/Human Motilin(GPR38) Stable Cell

SPECIES: Human

TARGET FAMILY: Motilin receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0157A


CHO-K1/Human MRGPRD Stable Cell

SPECIES: Human

TARGET FAMILY: MRGPRD

PARENTAL LINE: CHO-K1

ASSAY MODE: Calcium

CATALOG: SNB-G-0265A


CHO-K1/Human MRGPRX1 Stable Cell

SPECIES: Human

TARGET FAMILY: MRGPRX1

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0269D


HEK293/Human MRGPRX1 Stable Cell

SPECIES: Human

TARGET FAMILY: MRGPRX1

PARENTAL LINE: HEK293

ASSAY MODE: IP-1

CATALOG: SNB-G-0269A


HEK293/Human MRGPRX2 Stable Cell

SPECIES: Human

TARGET FAMILY: MRGPRX2

PARENTAL LINE: HEK293

ASSAY MODE: IP-1

CATALOG: SNB-G-0270D


CHO-K1/Human NMU1 Stable Cell

SPECIES: Human

TARGET FAMILY: NMU1 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0159A


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