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ScreeNingBio's GPCR Solution:
Assay Designed to Reach Your Goal Faster

​​Comprehensive GPCR Coverage

  • Ready-to use stable cell lines covering 80% GPCR drug targets

Native Expression Advantage

  • Full-length GPCRs stably expressed without artificial tags to preserve native receptor pharmacology

Flexible Assay Readouts

  • Multiple assay formats available, including cAMP, calcium flux, β-arrestin recruitment, IP-One, and reporter gene readouts, to meet diverse discovery needs

Cross-Species Capabilities

  • Broad panel of human, mouse, rat, dog, and cynomolgus monkey targets available for translational research

GPCR Family Tree.jpg
Target Receptors
按 类别-Target Receptors 篩選
Species
按 类别-Species 篩選
Assay Mode
按 类别-Assay Mode 篩選
Parental Line
按 类别-Receptor Form 篩選
CHO-K1/Mouse Glucagon Stable Cell

SPECIES: Mouse

TARGET FAMILY: Glucagon receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0105B


CHO-K1/Mouse Secretin Stable Cell

SPECIES: Mouse

TARGET FAMILY: Secretin receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0104B


CHO-K1/Rat GHRH Stable Cell

SPECIES: Rat

TARGET FAMILY: GHRH receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0102C


CHO-K1/Rat GIP Stable Cell

SPECIES: Rat

TARGET FAMILY: GIP receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0103C


CHO-K1/Rat GLP-1 Stable Cell

SPECIES: Rat

TARGET FAMILY: GLP-1 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0106C


CHO-K1/Rat GLP-2 Stable Cell

SPECIES: Rat

TARGET FAMILY: GLP-2 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0107C


CHO-K1/Rat Glucagon Stable Cell

SPECIES: Rat

TARGET FAMILY: Glucagon receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0105C


CHO-K1/Rat Secretin Stable Cell

SPECIES: Rat

TARGET FAMILY: Secretin receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0104C


HEK293/Dog GIPR Stable Cell

SPECIES: Dog

TARGET FAMILY: GIP receptor

PARENTAL LINE: HEK293

ASSAY MODE: cAMP

CATALOG: SNB-G-0103E


HEK293/Human GIP Stable Cell

SPECIES: Human

TARGET FAMILY: GIP receptor

PARENTAL LINE: HEK293

ASSAY MODE: cAMP

CATALOG: SNB-G-0103A


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