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ScreeNingBio's GPCR Solution:
Assay Designed to Reach Your Goal Faster

​​Comprehensive GPCR Coverage

  • Ready-to use stable cell lines covering 80% GPCR drug targets

Native Expression Advantage

  • Full-length GPCRs stably expressed without artificial tags to preserve native receptor pharmacology

Flexible Assay Readouts

  • Multiple assay formats available, including cAMP, calcium flux, β-arrestin recruitment, IP-One, and reporter gene readouts, to meet diverse discovery needs

Cross-Species Capabilities

  • Broad panel of human, mouse, rat, dog, and cynomolgus monkey targets available for translational research

GPCR Family Tree.jpg
Target Receptors
按 类别-Target Receptors 篩選
Species
按 类别-Species 篩選
Assay Mode
按 类别-Assay Mode 篩選
Parental Line
按 类别-Receptor Form 篩選
CHO-K1/Mouse FPR2-ALX Stable Cell

SPECIES: Mouse

TARGET FAMILY: FPR2-ALX

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0091B


HEK293T Human FPR3 β-Arrestin Stable Cell

SPECIES: Human

TARGET FAMILY: FPR3

PARENTAL LINE: HEK293T

ASSAY MODE: β-Arrestin

CATALOG: SNB-A-0092A



CHO-K1/Rat FFA4 (GPR120) Stable Cell

SPECIES: Rat

TARGET FAMILY: FFA4 receptor

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0096C


HEK293/Human FFA4 (GPR120) Stable Cell

SPECIES: Human

TARGET FAMILY: FFA4 receptor

PARENTAL LINE: HEK293

ASSAY MODE: IP-1

CATALOG: SNB-G-0096A


HEK293/Human FFA1(GPR40) Stable Cell

SPECIES: Human

TARGET FAMILY: FFAR1

PARENTAL LINE: HEK293

ASSAY MODE: IP-1

CATALOG: SNB-G-0093A


CHO-K1/Human FFA2 (GPR43) Stable Cell

SPECIES: Human

TARGET FAMILY: FFAR2

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0094A


CHO-K1/Human FFA3 (GPR41) Stable Cell

SPECIES: Human

TARGET FAMILY: FFAR3

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0095A


CHO-K1/Mouse FFA2 (GPR43) Stable Cell

SPECIES: Mouse

TARGET FAMILY: FFAR2

PARENTAL LINE: CHO-K1

ASSAY MODE: IP-1

CATALOG: SNB-G-0094B


CHO-K1/Mouse FFA3 (GPR41) Stable Cell

SPECIES: Mouse

TARGET FAMILY: FFAR3

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0095B


CHO-K1/Rat FFA3 (GPR41) Stable Cell

SPECIES: Rat

TARGET FAMILY: FFAR3

PARENTAL LINE: CHO-K1

ASSAY MODE: cAMP

CATALOG: SNB-G-0095C


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